Owner Exelixis Inc.

Inventors Chan, Diva Sze-Ming; Jones, Lisa Renee; Forsyth, Timothy Patrick; Rao, Pallavi; Chen, Jeff; Mac, Morrison B.; Franzini, Maurizio; Noguchi, Robin Tammie; Kelley, Ryan Michael; Jeong, Joon Won; Xu, Wei; Chan, Bryan; Leahy, James W.; Wang, Yong; Jammalamadaka, Vasu; Bahceci, Suleyman; Ridgway, Brian Hugh; Kim, Moon Hwan

Agent Davies Collison Cave

Pub. Number AU-A-2009266806

PCT Pub. Number WO2010/003133

Priority 61/134,047 03.07.08 US

Filing date 2 July 2009

Wipo publication date 7 January 2010

C07D 471/04 (2006.01) Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups

A61K 31/437 (2006.01)

A61K 31/506 (2006.01) - not condensed and containing further heterocyclic rings

A61K 31/519 (2006.01) - ortho- or peri-condensed with heterocyclic rings

A61K 31/5377 (2006.01)

A61K 31/5383 (2006.01)

A61K 31/55 (2006.01) - having seven-membered rings, e.g. azelastine, pentylenetetrazole

A61P 35/00 (2006.01) Antineoplastic agents

C07D 487/04 (2006.01) Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups

C07D 487/10 (2006.01) Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups

C07D 491/107 (2006.01) Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or

C07D 498/04 (2006.01) Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms

C07D 498/14 (2006.01) Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms