Owner Genentech, Inc. Curis, Inc.

Inventors Olivero, Alan G.; Lee, Wendy; Sutherlin, Daniel P.; Goldsmith, Richard A.; Robarge, Kirk D.

Agent Davies Collison Cave

Pub. Number AU-A-2006315467

PCT Pub. Number WO2007/059157

Priority 60/735,861 14.11.05 US

Filing date 14 November 2006

Wipo publication date 24 May 2007

C07D 213/82 (2006.01) Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members

A61K 31/167 (2006.01) - having the nitrogen atom of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol

A61K 31/4164 (2006.01) - 1,3-Diazoles

A61K 31/4196 (2006.01) - 1,2,4-Triazoles

A61K 31/44 (2006.01) - Non-condensed pyridines

A61K 31/444 (2006.01)

A61K 31/4453 (2006.01) - only substituted in position 1, e.g. propipocaine, diperodon

A61K 31/4545 (2006.01)

A61K 31/496 (2006.01) - Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene

A61K 31/5375 (2006.01) - 1,4-Oxazines, e.g. morpholine

C07D 231/14 (2006.01) Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings

C07D 239/28 (2006.01) Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings

C07D 277/56 (2006.01) Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings

C07D 401/12 (2006.01) Heterocyclic compounds containing two or more hetero rings

C07D 417/12 (2006.01) Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group