Owner Janssen Pharmaceutica N.V.

Inventors Santillan, Alejandro; Grice, Cheryl A.; Shaw, Karen J.; Hack, Michael D.; Gomez, Laurent; Wiener, John J.M.; Schwarz, Kimberly L.; Allison, Brett D.; Morrow, Brian J.; Venkatesan, Hariharan; Motley, Timothy S.; Tang, Liu Y.

Agent Shelston IP

Pub. Number AU-B-2006230364

PCT Pub. Number WO2006/105289

Priority 60/667,198 31.03.05 US

Filing date 30 March 2006

Wipo publication date 5 October 2006

Acceptance publication date 13 September 2012

C07D 221/02 Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups

A61K 31/44 - Non-condensed pyridines

A61K 31/47 - Quinolines

A61K 31/50 - Pyridazines

A61K 31/535 - having six-membered rings with at least one nitrogen and at least one oxygen as the ring hetero atoms, e.g. 1,2-oxazines

A61K 31/54 - having six-membered rings with at least one nitrogen and at least one sulfur as the ring hetero atoms, e.g. sulthiame

A61K 31/55 - having seven-membered rings, e.g. azelastine, pentylenetetrazole

C07D 279/12 Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms

C07D 413/00 Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms

C07D 417/00 Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group

C07D 471/00 Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups

C07D 471/02 Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups