Derivatives of N-(1H-indazolyl)- and N- (1H-indolyl)-urea as well as related compounds as modulators of the vanilloid-1 receptor (VR1) for the treatment of pain

Details for Australian Patent Application No. 2004274230 (hide)

Owner Merck Sharp & Dohme Limited

Inventors Fletcher, Stephen Robert; Rogers, Lauren; Jones, A. Brian; Moyes, Christopher Richard; Hollingworth, Gregory John

Agent Spruson & Ferguson

Pub. Number AU-A-2004274230

PCT Pub. Number WO2005/028445

Priority 0322016.7 19.09.03 GB

Filing date 16 September 2004

Wipo publication date 31 March 2005

International Classifications

A61K 31/416 (2006.01) - condensed with carbocyclic ring systems, e.g. indazole

A61K 31/343 (2006.01) - condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone

A61K 31/404 (2006.01)

A61K 31/4245 (2006.01) - Oxadiazoles

A61K 31/428 (2006.01) - condensed with carbocyclic rings

A61K 31/437 (2006.01)

C07C 275/28 (2006.01) Derivatives of urea, i.e. compounds containing any of the groups the nitrogen atoms not being part of nitro or nitroso groups

C07D 209/08 (2006.01) Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom

C07D 209/34 (2006.01) Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom

C07D 231/56 (2006.01) Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings

C07D 263/56 (2006.01) Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings

C07D 275/04 (2006.01) Heterocyclic compounds having nitrogen and sulfur as the only ring hetero atoms

C07D 277/62 (2006.01) Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings

C07D 307/79 (2006.01) Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom

C07D 471/04 (2006.01) Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups

Event Publications

9 March 2006 PCT application entered the National Phase

  PCT publication WO2005/028445 Priority application(s): WO2005/028445

14 August 2008 Application Lapsed, Refused Or Withdrawn, Patent Ceased or Expired

  This application lapsed under section 142(2)(a). A direction to request examination has been given for this application. Note that applications or patents shown as lapsed or ceased may be restored at a later date.

Legal

The information provided by the Site not in the nature of legal or other professional advice. The information provided by the Site is derived from third parties and may contain errors. You must make your own enquiries and seek independent advice from the relevant industry professionals before acting or relying on any information contained herein. Check the above data against the Australian Patent Office AUSPAT database.

Next and Previous Patents/Applications

2004274239-Polymorphic forms of a known antihyperlipemic agent

2004274227-Quinazoline derivatives