Owner Laboratoires Serono SA

Inventors Gerber, Patrick; Bombrun, Agnes; Swinnen, Dominique; Gonzalez, Jerome; Pittet, Pierre-Andre

Agent Griffith Hack

Pub. Number AU-B-2003239296

PCT Number PCT/EP03/00808

PCT Pub. Number WO2003/064376

Priority 02100078.1 29.01.02 EP; 02100410.6 25.04.02 EP

Filing date 27 January 2003

Wipo publication date 2 September 2003

Acceptance publication date 23 October 2008

C07C 237/42 (2006.01) Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups

A61K 31/198 (2006.01)

A61K 31/275 (2006.01) - Nitriles

A61K 31/343 (2006.01) - condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone

A61K 31/36 (2006.01)

A61K 31/381 (2006.01) - having five-membered rings

A61K 31/4245 (2006.01) - Oxadiazoles

A61K 31/426 (2006.01) - 1,3-Thiazoles

A61K 31/433 (2006.01) - Thiadiazoles

A61K 31/44 (2006.01) - Non-condensed pyridines

A61K 31/4402 (2006.01) - only substituted in position 2, e.g. pheniramine, bisacodyl

A61K 31/4409 (2006.01) - only substituted in position 4, e.g. isoniazid, iproniazid

A61K 31/4436 (2006.01)

A61K 31/445 (2006.01) - Non-condensed piperidines, e.g. piperocaine

A61K 31/498 (2006.01) - Pyrazines or piperazines ortho- or peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine

A61K 31/5377 (2006.01)

A61K 45/00 (2006.01) Medicinal preparations containing active ingredients not provided for in groups

A61P 3/04 (2006.01) Drugs for disorders of the metabolism

A61P 3/06 (2006.01) Drugs for disorders of the metabolism

A61P 3/10 (2006.01) Drugs for disorders of the metabolism

A61P 15/00 (2006.01) Drugs for genital or sexual disorders

A61P 43/00 (2006.01) Drugs for specific purposes, not provided for in groups

C07B 61/00 (2006.01) Other general methods