Owner ELI LILLY AND COMPANY

Inventors Xie, Chaoyu; Biggers, Christopher, Kelly; Doecke, Christopher, William; Shah, Jikesh, Arvind; Mayer, John, Philip; Briner, Karin; Wu, Zhipei; Fisher, Matthew, Joseph; Martinelli, Michael, John; Ornstein, Paul, Leslie; Shi, Qing; Richardson, Timothy, Ivo; Mancoso, Vincent; Hertel, Larry, Wayne

Agent Spruson & Ferguson

Pub. Number AU-A-2002246969

PCT Pub. Number WO2002/059108

Priority 60/263,471 23.01.01 US

Filing date 23 January 2002

Wipo publication date 6 August 2002

C07D 401/12 Heterocyclic compounds containing two or more hetero rings

C07D 403/12 Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group

C07D 409/14 Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms

A61K 031/495 - having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine

A61K 031/535 - having six-membered rings with at least one nitrogen and at least one oxygen as the ring hetero atoms, e.g. 1,2-oxazines

A61K 031/55 - having seven-membered rings, e.g. azelastine, pentylenetetrazole

A61P 003/00 Drugs for disorders of the metabolism

A61P 015/00 Drugs for genital or sexual disorders

C07D 403/14 Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group

C07D 401/14 Heterocyclic compounds containing two or more hetero rings

C07D 413/14 Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms

C07D 417/14 Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group